PXS-4787 hydrochloride

SKU: orb2695237

Description

PXS-4787 hydrochloride is a specific and potent pan-lysyl oxidase inhibitor that effectively eliminates the activity of lysyl oxidase. It exhibits varying IC50 values against different forms of the enzyme, including 2 μM (Bovine LOX), 3.2 μM (rh LOXL1), 0.6 μM (rh LOXL2), 1.4 μM (rh LOXL3), and 0.2 μM (rh LOXL4). In addition, PXS-4787 hydrochloride reduces the deposition and cross-linking of collagen I secreted by human fibroblasts.

Research Area

,Neuroscience

Key Properties

• CAS Number: 2409964-40-3
• MW: 265.73
• Formula: C₁₀H₁₃ClFNO₂S
• SMILES: S(C/C(=C/CN)/F)(=O)(=O)C1=CC=CC=C1.Cl

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

68770906