RGB286638

SKU: orb251372

Description

RGB-286638 is a novel CDK inhibitor with IC50s of 1 nM/2 nM/3 nM/4 nM/5 nM for cyclin T1-CDK9/cyclin B1-CDK1/cyclin E-CDK2/cyclin D1-CDK4/cyclin E-CDK3/p35-CDK5 respectively; less potent against cyclin H-CDK7 and cyclin D3-CDK6.

Research Area

Product Categories/Products/Small Molecules

Key Properties

• CAS Number: [784210-88-4]
• MW: 545.64
• Formula: C₂₉H₃₅N₇O₄
• SMILES: N(C1=CC=CC2C3=C(C(=O)C1=2)C(C1=CC=C(CN2CCN(CCOC)CC2)C=C1)=NN3)C(NN1CCOCC1)=O

Storage & Handling

• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only